MK 1256

Overview

MK 1256 is a highly selective and orally active inhibitor of tissue protease K ( Cat K ) with an IC 50 of 0.62 nM. MK 1256 shows extremely high selectivity towards other tissue proteases (all > 1100 times), with only a slightly lower selectivity for tissue protease F (Cat F) (110 times). MK 1256 exhibits strong anti-bone resorption activity in the osteoporosis model of rhesus monkeys with ovariectomy. MK 1256 can be used for research on osteoporosis.

Application

Products | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Metabolic Disease | Products > Signaling Pathways > Cathepsin

Product Information

• Catalog No.: HY-14360
• CAS No.: 919109-76-5
• Molecular Formula: C23H23Cl2F3N4O3S
• Molecular Weight: 563.42
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source