MS5033 is a potent PROTAC-based AKT (protein kinase B) degrader, with a DC 50 of 430 nM in PC3 cells. (Pink: Akt ligand ( HY-48682 ); Blue: Cereblon ligand ( HY-10984 ); Black: linker ( HY-133051 )).
Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > PI3K/Akt/mTOR | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > Akt
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