Talarozole

Overview

Talarozole (R115866) is an oral systemic all-trans retinoic acid metabolism blocking agent (RAMBA) which increases intracellular levels of endogenous all-trans retinoic acid (RA). Talarozole inhibits both CYP26A1 and CYP26B1 with IC 50 s of 5.4 and 0.46 nM, respectively.

Application

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Product Information

• Catalog No.: HY-14531
• CAS No.: 201410-53-9
• Molecular Formula: C21H23N5S
• Molecular Weight: 377.51
• Purity: 99.75%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2 mg/mL (5.30 mM); Suspended solution
• Availability: In-stock

Source

Original product source