Desmethyl Bosentan

Overview

Desmethyl bosentan is an active metabolite of the endothelin receptor antagonist bosentan ( HY-A0013 ).1 Desmethyl bosentan (25 μM) activates the pregnane X receptor (PXR) in CV-1 monkey kidney cells expressing the human receptor in a reporter assay.

Application

Products | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Metabolic Disease | Products > Signaling Pathways > Drug Metabolite | Products > Signaling Pathways > Cytochrome P450

Product Information

• Catalog No.: HY-145516
• CAS No.: 253688-61-8
• Molecular Formula: C26H27N5O6S
• Molecular Weight: 537.59
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source