Tyrphostin AG 528

Tyrphostin AG 528
  • CAS No.:133550-49-9
  • Grade:98.0%
  • Formula:C18H14N2O3
  • M.W.:306.32
  • Solvent:≥ 2.5 mg/mL (8.16 mM); Clear solution

Overview

Tyrphostin AG 528 is an inhibitor of EGFR and ErbB2 with IC 50 s of 4.9 and 2.1 μM, respectively. Tyrphostin AG 528 (Tyrphostin B66) is a protein tyrosine kinase inhibitor, with IC 50 s of 4.9 μM for epidermal growth factor receptors ( EGFR ) and 2.1 μM for ErbB2 . Tyrphostin AG 528 is also an anticancer agent.

Application

Products | Products > Disease Areas > Hepatitis Virus Infection | Products > Disease Areas > Lipid Metabolism | Products > Disease Areas > Lung Cancer | Products > Disease Areas > Breast Cancer | Products > Disease Areas > Colorectal Cancer | Products > Disease Areas > Digestive System Cancer | Products > Disease Areas > Prostate Cancer | Products > Disease Areas > Urogenital Cancer | Products > Disease Areas > Gastric Cancer | Products > Disease Areas > Liver Cancer | Products > Disease Areas > Pancreatic Cancer | Products > Disease Areas > Ovarian Cancer | Products > Disease Areas > Hepatitis C Virus Infection | Products > Disease Areas > Obesity | Products > Disease Areas > Cancer | Products > Disease Areas > Infection | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Disease Areas > Digestive System Disease | Products > Disease Areas > Urogenital Disease | Products > Signaling Pathways > JAK/STAT Signaling | Products > Signaling Pathways > Protein Tyrosine Kinase/RTK | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > EGFR

Product Information

  • Catalog No.: HY-100499
  • CAS No.: 133550-49-9
  • Molecular Formula: C18H14N2O3
  • Molecular Weight: 306.32
  • Purity: 98.0%
  • Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
  • Solubility: ≥ 2.5 mg/mL (8.16 mM); Clear solution
  • Availability: In-stock

Source

Original product source


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