Rosiglitazone maleate

Overview

Rosiglitazone maleate (BRL 49653C) is a potent and selective activator of PPARγ , with EC 50 s of 30 nM, 100 nM and 60 nM for PPARγ1 , PPARγ2 , and PPARγ , respectively, and a K d of appr 40 nM for PPARγ ; Rosiglitazone maleate is also an modulator of TRP channels , inhibits TRP melastatin 2 (TRPM2), TRPM3 and activates TRP canonical 5 (TRPC5).

Application

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Product Information

• Catalog No.: HY-14600
• CAS No.: 155141-29-0
• Molecular Formula: C22H23N3O7S
• Molecular Weight: 473.50
• Purity: 99.73%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.5 mg/mL (5.28 mM); Clear solution
• Availability: In-stock

Source

Original product source