PqsR/LasR-IN-1 (compound 2a) is a potent PqsR and LasR systems inhibitor. PqsR/LasR-IN-1 has anti-virulence activity against Pseudomonas aeruginosa . PqsR/LasR-IN-1 can reduce production of biofilm, pyocyanin, and rhamnolipids in PA.
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