FAAH/MAGL-IN-3 (Compound 10) is an irreversible fatty acid amide hydrolase ( FAAH ) and monoacylglycerol lipase ( MAGL ) dual inhibitor with IC 50 values of 179 and 759 nM against FAAH and MAGL , respectively. FAAH/MAGL-IN-3 shows low PAMPA (Parallel Artificial Membrane Permeability Assay) permeability.
Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > FAAH | Products > Signaling Pathways > MAGL
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