PROTAC CYP1B1 degrader-1 is a CYP1B1 PROTAC degrader with a human IC 50 of 95.1 nM. PROTAC CYP1B1 degrader-1 induces concentration-dependent CYP1B1 degradation. PROTAC CYP1B1 degrader-1 can be used for the research of CYP1B1 -mediated Docetaxel ( HY-B0011 )-resistant prostate cancer . (Pink: CYP1B1 Target protein ligand; Blue: Cereblon ligand ( HY-103596 ); Black: linker).
Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Drug Resistance | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > Cytochrome P450
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