BMY 7378

Overview

BMY 7378 is a selective antagonist of α 1D -adrenoceptor (α 1D -AR). BMY 7378 binds to membranes expressing the cloned rat α 1D -AR with a >100-fold higher affinity ( K i =2 nM) than binding to either the cloned rat α 1A -AR (K i =800 nM) or the hamster α 1B -AR ( K i =600 nM). BMY 7378 is a 5-HT 1A receptor partial agonist.

Application

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Product Information

• Catalog No.: HY-100554
• CAS No.: 21102-95-4
• Molecular Formula: C22H33Cl2N3O3
• Molecular Weight: 458.42
• Purity: 99.92%
• Storage: 4°C, sealed storage, away from moisture and light * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
• Solubility: ≥ 5 mg/mL (10.91 mM); Clear solution
• Availability: In-stock

Source

Original product source