PF-07258669

Overview

PF-07258669 is an orally active melanocortin-4 receptor ( MC4R ) antagonist that antagonizes MC4R with an IC 50 of 13 nM ( K i =0.46 nM). PF-07258669 can be used for the research of cachexia, anorexia, or anorexia nervosa.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Research Areas > Metabolic Disease | Products > Signaling Pathways > Melanocortin Receptor

Product Information

• Catalog No.: HY-148349
• CAS No.: 2755890-53-8
• Molecular Formula: C25H27FN6O2
• Molecular Weight: 462.52
• Purity: 98.44%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (5.41 mM); Clear solution
• Availability: In-stock

Source

Original product source