Akt1&PKA-IN-1 is a potent dual Akt/PKA inhibitor with IC 50 values of 0.03 , 0.11 μM, and 9.8 μM for PKAa, Akt , and CDK2 , respectively. Akt1&PKA-IN-1 is selective for cyclin-dependent kinase 2 (CDK2) .
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