3-Hydroxy darifenacin is a metabolite of Darifenacin ( HY-A0033 ). 3-Hydroxy darifenacin is an antagonist of M 1-5 muscarinic receptors with Kis values of 17.78, 79.43, 2.24, 36.31 and 6.17 nM, respectively in CHO cells.
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