VUF11207 (Compound 29) is a CXCR7 agonist and a high-potency CXCR7 ( pK i of 8.1) ligand that induces recruitment of β-arrestin2 ( pEC 50 of 8.8) and subsequent internalization ( pEC 50 of 7.9) of CXCR7 .
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