CHF-6366 is a potent M3 muscarinic antagonist and β2-adrenergic receptors agonist with pK i values of 10.4 and 11.4, respectively. CHF-6366 is also a weak calcium channel inhibitor ( IC 50 ~50 μM). CHF-6366 inhibits bronchoconstriction in guinea pigs. CHF-6366 can be used to research chronic obstructive pulmonary disease (COPD).
Products | Products > Disease Areas > Inflammation or Immune System Disease | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Research Areas > Inflammation/Immunology | Products > Research Areas > Endocrinology | Products > Signaling Pathways > mAChR | Products > Signaling Pathways > Adrenergic Receptor | Products > Signaling Pathways > Calcium Channel
感谢您来到爆牛贸易,请为我们留言或者使用以下方式联系我们,我们将尽快给您回复,并为您提供最真诚的服务,谢谢。