SIAIS100 is a potent BCR-ABL PROTAC degrader with an DC 50 value of 2.7 nM. SIAIS100 can be used to research chronic myeloid leukemia (CML). (Pink: Target protein ligand; Blue: Cereblon ligand ( HY-W586108 ); Black: linker).
Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > Protein Tyrosine Kinase/RTK | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > Bcr-Abl
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