GS-6201 (Standard)

Overview

GS-6201 (Standard) is the analytical standard of GS-6201 ( HY-10081 ). This product is intended for research and analytical applications. GS-6201 (CVT-6883) is a selective adenosine A2B receptor antagonist. GS-6201 displays high affinity and selectivity for the human adenosine A2B receptors (Ki=22 nM). GS-6201 reduces caspase-1 activity in the heart, and attenuates cardiac remodeling after acute myocardial infarction (AMI) in the mouse. GS-6201 3 attenuates the airway reactivity induced by NECA, AMP, or allergen in sensitized mice.

Application

Products | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Others | Products > Research Areas > Inflammation/Immunology | Products > Signaling Pathways > Adenosine Receptor | Products > Signaling Pathways > Reference Standards

Product Information

• Catalog No.: HY-10081R
• CAS No.: 752222-83-6
• Molecular Formula: C21H21F3N6O2
• Molecular Weight: 446.43
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source