RS-127445 hydrochloride

Overview

RS-127445 hydrochloride is a selective, high affinity, orally bioavailable 5-HT 2B receptor antagonist with a pK i of 9.5. RS-127445 hydrochloride shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites.

Application

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Product Information

• Catalog No.: HY-15419
• CAS No.: 199864-86-3
• Molecular Formula: C17H17ClFN3
• Molecular Weight: 317.79
• Purity: 99.78%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.5 mg/mL (7.87 mM); Clear solution
• Availability: In-stock

Source

Original product source