PROTAC TG2 degrader-1

PROTAC TG2 degrader-1
  • CAS No.:3033465-55-0
  • Grade:99.98%
  • Formula:C55H73N9O10S
  • M.W.:1052.29

Overview

PROTAC TG2 degrader-1 (compound 11) is a von Hippel-Lindau (VHL)-based PROTAC targeting tissue transglutaminase (TG2) with a K D of 68.9 μM. PROTAC TG2 degrader-1 reduces TG2 in ovarian cancer cells in a proteasome-dependent manner.

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > Glutaminase

Product Information

  • Catalog No.: HY-155643
  • CAS No.: 3033465-55-0
  • Molecular Formula: C55H73N9O10S
  • Molecular Weight: 1052.29
  • Purity: 99.98%
  • Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source


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