HA-100 (Standard) is the analytical standard of HA-100 ( HY-100984 ). This product is intended for research and analytical applications. HA-100 is a potent protein kinase inhibitor, with IC50s of 4 μM, 8 μM, 12 μM and 240 μM for cGMP-dependent protein kinase ( PKG ), cAMP-dependent protein kinase ( PKA ), protein kinase C ( PKC ) and MLC-kinase, respectively. HA-100 also used as a ROCK inhibitor .
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