GSK4028

Overview

GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC 50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.

Application

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Product Information

• Catalog No.: HY-101027A
• CAS No.: 2079886-19-2
• Molecular Formula: C17H21BrN4O
• Molecular Weight: 377.28
• Purity: 98.06%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (6.63 mM); Clear solution
• Availability: In-stock

Source

Original product source