Rociletinib hydrobromide

Overview

Rociletinib hydrobromide (CO-1686 hydrobromide) is an orally delivered kinase inhibitor that specifically targets the mutant forms of EGFR including T790M, and the K i values for EGFRL858R/T790M and EGFRWT are 21.5 nM and 303.3 nM, respectively.

Application

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Product Information

• Catalog No.: HY-15729A
• CAS No.: 1446700-26-0
• Molecular Formula: C27H29BrF3N7O3
• Molecular Weight: 636.46
• Purity: 98.04%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.5 mg/mL (3.93 mM); Clear solution
• Availability: In-stock

Source

Original product source