5-HT2CR agonist 1

Overview

5-HT2CR agonist 1 (compound 8), a 7-chloro analogue, is a selective 5-HT 2C R partial agonist (E max =71.09%) with an EC 50 value of 121.5 nM and no observed activity toward 5-HT 2A R or 5-HT 2B R. 5-HT2CR agonist 1 exhibits no recruitment activity for β-arrestin and shows low inhibition of hERG at 10 μM.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > 5-HT Receptor

Product Information

• Catalog No.: HY-157425
• CAS No.: 1216074-15-5
• Molecular Formula: C13H14ClNO
• Molecular Weight: 235.71
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source