Aprocitentan (Standard)

Overview

Aprocitentan (Standard) is the analytical standard of Aprocitentan. This product is intended for research and analytical applications. Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively.

Application

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Product Information

• Catalog No.: HY-15895R
• CAS No.: 1103522-45-7
• Molecular Formula: C16H14Br2N6O4S
• Molecular Weight: 546.19
• Purity: 98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source