Aprocitentan-d 4

Overview

Aprocitentan-d 4 is a deuterium labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is an orally active dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively. Aprocitentan is an antihypertensive agent.

Application

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Product Information

• Catalog No.: HY-15895S
• CAS No.: 2748196-51-0
• Molecular Formula: C16H10D4Br2N6O4S
• Molecular Weight: 550.22
• Purity: 98.76%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Availability: In-stock

Source

Original product source