K-Opioid receptor agonist-1

Overview

K-Opioid receptor agonist-1 (Compound 5a) is an agonist for κ-Opioid receptor with K i of 0.25 nM and EC 50 of 2 nM. K-Opioid receptor agonist-1 is blood brain barrier (BBB) penetrate (brain/plasma ratios of 0.50 to 0.65). K-Opioid receptor agonist-1 exhibits anti-inflammatory activity in dermatitis models induced by Arachidonic acid ( HY-109590 ) or oxazolidinone .

Application

Products | Products > Disease Areas > Inflammation or Immune System Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Inflammation/Immunology | Products > Signaling Pathways > Opioid Receptor

Product Information

• Catalog No.: HY-160761
• CAS No.: 1816990-29-0
• Molecular Formula: C22H29Cl2N3O3
• Molecular Weight: 454.39
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source