uPSEM792

Overview

uPSEM792 is a pharmacologically selective effector molecules (PSEM) agonist for PSAM 4 -GlyR, with an affinity of K i of 0.7 nM. uPSEM792 is a substrate for efflux transporters in brains of wild type and dual P-gp and BCRP knockout mice. uPSEM7952 is a possible lead for developing the PET radioligand for PSAM 4 -GlyR.

Application

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Product Information

• Catalog No.: HY-161246
• CAS No.: 2323525-19-3
• Molecular Formula: C14H15N3O
• Molecular Weight: 241.29
• Purity: 98.02%
• Storage: 4°C, protect from light * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
• Solubility: ≥ 9.5 mg/mL (39.37 mM); Clear solution
• Availability: In-stock

Source

Original product source