CBP/p300 ligand 4 (Compound 4) is an orally active inhibitor for CBP/p300 bromodomain, with IC 50 of 91.4 nM. CBP/p300 ligand 4 serves as a ligand for target protein XYD190 ( HY-161495 ). XYD190 is a PROTAC degrader for CBP/p300 .
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