MYC degrader 1

Overview

MYC degrader 1 (compound A80.2HCl) is an orally available MYC molecular glues degrader with anti-tumor activity. MYC degrader 1 restores pRB1 protein activity and re-establishes sensitivity of MYC overexpressing cancer cells to CDK4/6 inhibitors.

Application

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Product Information

• Catalog No.: HY-162318
• CAS No.: 2946670-96-6
• Molecular Formula: C32H31ClF3N5O3
• Molecular Weight: 626.07
• Purity: 99.61%
• Storage: -20°C, sealed storage, away from moisture and light * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
• Solubility: ≥ 2.5 mg/mL (3.99 mM); Clear solution
• Availability: In-stock

Source

Original product source