σ1 Receptor/μ Opioid receptor modulator 2

Overview

σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/ σ1R antagonist, and displays picomolar μOR agonism activity ( EC 50 : 0.6 ± 0.2 nM) and good σ1R inhibitory activity ( K i : 363.7 ± 5.6 nM). σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > Opioid Receptor | Products > Signaling Pathways > Sigma Receptor

Product Information

• Catalog No.: HY-163065
• CAS No.: 3009018-61-2
• Molecular Formula: C23H31N3O
• Molecular Weight: 365.51
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source