VU 6008667

Overview

VU 6008667 is a selective negative allosteric modulator of M5 NAM with IC 50 s of 1.2 μM and 1.6 μM for human M5 and rat M5, respectively. High CNS penetration.

Application

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Product Information

• Catalog No.: HY-101281
• CAS No.: 2092923-21-0
• Molecular Formula: C24H17ClF2N2O2
• Molecular Weight: 438.85
• Purity: 99.53%
• Storage: 4°C, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
• Solubility: ≥ 2.5 mg/mL (5.70 mM); Clear solution
• Availability: In-stock

Source

Original product source