BRD4 degrader-2

Overview

BRD4 degrader-2 (Compound JP-2-197) is a covalent monovalent molecular glue BRD4 degrader that induces a ternary complex formation between BRD4 and RNF126. BRD4 degrader-2 targets RNF126 (E3 ligase ) and degrades both the long and short isoforms of BRD4 in cells.

Application

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Product Information

• Catalog No.: HY-163639
• CAS No.: 3036530-43-2
• Molecular Formula: C34H33ClN6O4S
• Molecular Weight: 657.18
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source