CDK2 degrader 2

CDK2 degrader 2
  • CAS No.:3030271-16-7
  • Grade:99.51%
  • Formula:C46H57ClN10O6S
  • M.W.:913.53

Overview

CDK2 degrader 2 (Compound I-10) is a PROTAC degrader for CDK2 that degrades CDK2 in MKN1 cell with a DC 50 <100 nM. (Pink: CDK2 ligand ( HY-176124 ); Blue: Cereblon ligand ( HY-45512 ); Black: linker ( HY-W687952 )).

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > CDK

Product Information

  • Catalog No.: HY-163815
  • CAS No.: 3030271-16-7
  • Molecular Formula: C46H57ClN10O6S
  • Molecular Weight: 913.53
  • Purity: 99.51%
  • Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
  • Availability: In-stock

Source

Original product source


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