PROTAC HDAC8 Degrader-1

PROTAC HDAC8 Degrader-1
  • CAS No.:3057302-08-3
  • Grade:99.98%
  • Formula:C32H44N6O4
  • M.W.:576.73

Overview

Degrader-1 (compound Z16) is a potent and selective HDAC8 PROTAC degrader with an DC 50 of 0.27 nM in A549 cells. (Pink: HDAC8 ligand ( HY-163921 ); Blue: Cereblon ligand ( HY-150799 ); Black: linker).

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Signaling Pathways > Epigenetics | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > HDAC

Product Information

  • Catalog No.: HY-163920
  • CAS No.: 3057302-08-3
  • Molecular Formula: C32H44N6O4
  • Molecular Weight: 576.73
  • Purity: 99.98%
  • Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source


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