GW9662-d 5 is the deuterium labeled GW9662. GW9662 is a potent and selective PPARγ antagonist with an IC 50 of 3.3 nM, showing 10 and 1000-fold selectivity over PPARα and PPARδ , respectively.
Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Others | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Signaling Pathways > Vitamin D Related/Nuclear Receptor | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Signaling Pathways > Isotope-Labeled Compounds | Products > Signaling Pathways > PPAR
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