Famlasertib

Overview

Famlasertib is a potent, brain-penetrant MAP4K inhibitor with IC 50 s value of 0.3 nM, 23.7 nM, and 44.7 nM for HGK (MAP4K4), MLK3, and MLK1, respectively. Famlasertib shows motor neuron protection and anti-inflammatory properties. Famlasertib can be used for the study of amyotrophic lateral sclerosis (ALS).

Application

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Product Information

• Catalog No.: HY-168972
• CAS No.: 2375591-69-6
• Molecular Formula: C26H27ClN4O
• Molecular Weight: 446.97
• Purity: 99.94%
• Storage: 4°C, protect from light * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
• Solubility: 5 mg/mL (11.19 mM); Suspended solution; Need ultrasonic
• Availability: In-stock

Source

Original product source