ARV-825

Overview

ARV-825 is a PROTAC connected by ligands for Cereblon and BRD4 . ARV-825 binds to BD1 and BD2 of BRD4 with K d s of 90 and 28 nM, respectively.

Application

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Product Information

• Catalog No.: HY-16954
• CAS No.: 1818885-28-7
• Molecular Formula: C46H47ClN8O9S
• Molecular Weight: 923.43
• Purity: 99.21%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 1 year , -20°C, 6 months
• Solubility: ≥ 2.5 mg/mL (2.71 mM); Clear solution
• Availability: In-stock

Source

Original product source