Vicriviroc maleate

Overview

Vicriviroc maleate (SCH-417690 maleate; SCH-D maleate) is a potent, selective, oral bioavailable and CNS penetrated antagonist of CCR5 , with a K i of 2.5 nM, and also inhibits HIV-1 in PBMC cells, with IC 90 s of 3.3 nM (JrFL), 2.8 nM (ADA-M), 1.8 nM (301657), 4.9 nM (JV1083) and 10 nM (RU 570).

Application

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Product Information

• Catalog No.: HY-17377
• CAS No.: 599179-03-0
• Molecular Formula: C32H42F3N5O6
• Molecular Weight: 649.70
• Purity: 98.49%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.5 mg/mL (3.85 mM); Clear solution
• Availability: In-stock

Source

Original product source