Rosiglitazone -d 4 is deuterated labeled Rosiglitazone ( HY-17386 ). Rosiglitazone (BRL 49653) is an orally active selective PPARγ agonist ( EC 50 : 60 nM, K d : 40 nM). Rosiglitazone is an TRPC5 activator ( EC 50 : 30 μM) and TRPM3 inhibitor. Rosiglitazone can be used in the research of obesity and diabetes, senescence, ovarian cancer .
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