PI4Kβ/PKG-IN-2 (Compound 20) is an orally active dual inhibitor of Plasmodium phosphatidylinositol 4-kinase beta ( PI4Kβ ) and cGMP-dependent protein kinase ( PKG ). PI4Kβ/PKG-IN-2 has potent inhibitory effects on Plasmodium . PI4Kβ/PKG-IN-2 is promising for research of malaria.
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