PROTAC HDAC6 degrader 6 (Compound 12) is a selective HDAC6 -targeting photochemically targeting chimeras (PHOTACs) (subset of PROTAC ) degrader with a ~50% D max only upon activation to its cis -state with 390 nm light irradiation. (Pink: Target protein ligand; Blue: Cereblon ligand ( HY-A0003 ); Black: linker).
Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > Epigenetics | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > HDAC
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