Olaparib -d 4 -1 (AZD2281-d 4 -1) is the deuterium labeled Olaparib ( HY-10162 ). Olaparib is a potent and orally active PARP inhibitor with IC 50 s of 5 and 1 nM for PARP1 and PARP2 , respectively. Olaparib is an autophagy and mitophagy activator .
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