PROTAC PDIA1 degrader 1 (Compound H4) is a PDIA1 PROTAC degrader with a DC 50 of 29.71 μM. PROTAC PDIA1 degrader 1 has potent anticancer activity and significantly inhibits cancer cell proliferation. Pink: PDIA1 ligand ( HY-100433 ); Blue: CRBN ligase ligand ( HY-10984 ); Black: linker ( HY-W015088 ) (Pink: PDIA1 ligand ( HY-100433 ); Blue: Cereblon ligand ( HY-10984 ); Black: linker ( HY-W015088 )).
Products | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > PDI
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