SERT/5-HT-IN-1

Overview

SERT/5-HT-IN-1 (compound D17) is an orally active and potent dual target inhibitor of SERT/5-HT3A ( SERT IC 50 = 1.5 nM, NET IC 50 = 49 nM, DAT IC 50 = 91 nM, 5-HT3A K i = 12 nM). SERT/5-HT-IN-1 has an IC 50 of 39 nM to 5-HT3A. SERT/5-HT-IN-1 has a lower risk of liver, kidney, and cardiac toxicity. SERT/5-HT-IN-1 can be used for research on depressive disorders.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Disease Areas > Depression | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > GPCR/G Protein | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > Serotonin Transporter | Products > Signaling Pathways > 5-HT Receptor

Product Information

• Catalog No.: HY-178907
• CAS No.: 3120534-54-2
• Molecular Formula: C15H18N2S
• Molecular Weight: 258.38
• Purity: 99.44%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Availability: In-stock

Source

Original product source