Roluperidone

Overview

Roluperidone (CYR-101) is a novel cyclic amide derivative that has high equipotent affinities for 5-HT 2A and sigma-2 receptors ( K i of 7.53 nM and 8.19 nM for 5-HT 2A and sigma-2, respectively).

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > 5-HT Receptor | Products > Signaling Pathways > Sigma Receptor

Product Information

• Catalog No.: HY-19469
• CAS No.: 359625-79-9
• Molecular Formula: C22H23FN2O2
• Molecular Weight: 366.43
• Purity: 99.86%
• Storage: Powder -20°C, 3 years , 4°C, 2 years * The compound is unstable in solutions, freshly prepared is recommended.
• Solubility: ≥ 3 mg/mL (8.19 mM); Clear solution
• Availability: In-stock

Source

Original product source