DA-6886 monohydrochloride

Overview

DA-6886 is a 5-Hydroxytryptamine receptor 4 ( 5-HT4 ) agonist. DA-6886 induces relaxation of the rat oesophagus preparation in a 5-HT4 receptor antagonist-sensitive manner. The evaluation of DA-6886 in CHO cells expressing hERG channels reveals that it inhibits hERG channel current with an pIC 50 value of 4.3, indicating that the compound is 1000-fold more selective for the 5-HT4 receptor over hERG channels. DA-6886 can be used in the study of constipated irritable bowel syndrome.

Application

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Product Information

• Catalog No.: HY-19927A
• CAS No.: 1645260-76-9
• Molecular Formula: C19H28Cl2N6O2
• Molecular Weight: 443.37
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source