GSK137647A

Overview

GSK137647A (GSK 137647) is a potent, selective free fatty acid receptor 4 ( FFA4 ) agonist with pEC 50 values of 6.3, 6.2, and 6.1 for human, mouse and rat FFA4, and pEC 50 values < 4.5 for all three species for FFA1, FFA2, and FFA3, respectively. GSK137647A has anti-inflammatory activity. GSK137647A induces insulin secretion and inhibits epithelial ion transport, GSK137647A is related to regulation of glucose homeostasis and anti-inflammatory response.

Application

Products | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Research Areas > Metabolic Disease | Products > Signaling Pathways > Free Fatty Acid Receptor

Product Information

• Catalog No.: HY-19995
• CAS No.: 349085-82-1
• Molecular Formula: C16H19NO3S
• Molecular Weight: 305.39
• Purity: 99.81%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (8.19 mM); Clear solution
• Availability: In-stock

Source

Original product source