Lapatinib ditosylate monohydrate

Overview

Lapatinib ditosylate monohydrate (GW572016 ditosylate monohydrate) is a potent, orally active inhibitor of the ErbB-2 and EGFR tyrosine kinase domains with IC 50 values against purified EGFR and ErbB-2 of 10.2 and 9.8 nM, respectively.

Application

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Product Information

• Catalog No.: HY-50898B
• CAS No.: 388082-78-8
• Molecular Formula: C43H44ClFN4O11S3
• Molecular Weight: 943.48
• Purity: 99.99%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: 2.5 mg/mL (2.65 mM); Suspended solution; Need ultrasonic
• Availability: In-stock

Source

Original product source