SB-408124

SB-408124
  • CAS No.:288150-92-5
  • Grade:98.93%
  • Formula:C19H18F2N4O
  • M.W.:356.37
  • Solvent:≥ 2.5 mg/mL (7.02 mM); Clear solution

Overview

SB-408124 is a non-peptide OX1 receptor antagonist with K i s of 57 nM and 27 nM in whole cell and membrane, respectively. SB-408124 exhibits 50-fold selectivity over OX2 receptor.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Research Areas > Endocrinology | Products > Signaling Pathways > Orexin Receptor (OX Receptor)

Product Information

  • Catalog No.: HY-70068
  • CAS No.: 288150-92-5
  • Molecular Formula: C19H18F2N4O
  • Molecular Weight: 356.37
  • Purity: 98.93%
  • Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
  • Solubility: ≥ 2.5 mg/mL (7.02 mM); Clear solution
  • Availability: In-stock

Source

Original product source


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