Midostaurin-d 5 (PKC412-d 5 ) is a deuterium labeled Midostaurin. Midostaurin is a multi-targeted protein kinase inhibitor which inhibits PKCα/β/γ, Syk , Flk-1, Akt , PKA , c-Kit , c-Fgr, c-Src, FLT3 , PDFRβ and VEGFR1/2 with IC 50 s ranging from 22-500 nM.
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